Search references for SRX251. Phrases containing SRX251
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Pharmaceutical compound
SRX251, or SRX-251, also known as API-251, is a selective vasopressin V1A receptor antagonist that is or was under development for the treatment of aggression
SRX251
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
NTX-1472
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
SRX246
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Lithium_carbonate
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
LIT-002
Mammalian hormone released from the pituitary gland
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin
Peptide hormone and neuropeptide
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Oxytocin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Nelivaptan
Medication
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Desmopressin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Demeclocycline
Medication used for preventing postpartum bleeding
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Carbetocin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Tolvaptan
(MAO-B) inhibitor KNX-101 – 15-lipoxygenase (15-LOX; ALOX15) inhibitor SRX251 – vasopressin V1A receptor antagonist – no recent development since 2007
List of investigational aggression drugs
List_of_investigational_aggression_drugs
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
PF-184563
Agent that interferes with action at the vasopressin receptors
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin receptor antagonist
Vasopressin_receptor_antagonist
Medication causing uterine contraction
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Uterotonic
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
TGOT
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Oxytocin_receptor_agonist
Small-molecule oxytocin receptor agonist
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
LIT-001
Medication made from the peptide oxytocin
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Oxytocin_(medication)
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Terlipressin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Retosiban
Protein-coding gene in the species Homo sapiens
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin_receptor_2
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Barusiban
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Cligosiban
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Atosiban
Cleavage product of the coding protein of OXT gene
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Neurophysin_I
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
L-368,899
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasotocin
Carrier protein for oxytocin and vasopressin
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Neurophysins
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Lixivaptan
Type of drug that reduces aggression
Izenwasser S (eds.). "Orally active vasopressin V1a receptor antagonist, SRX251, selectively blocks aggressive behavior". Pharmacology, Biochemistry, and
Serenic
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Ornipressin
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
CA7_(drug)
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
TC_OT_39
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin_(medication)
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
WAY-267464
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Conivaptan
Genes on human chromosome 3
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Oxytocin_receptor
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Epelsiban
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
PF-06655075
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
L-371,257
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Selepressin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Demoxytocin
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Brezivaptan
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
NP-1031
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
WJ0679
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
KNX-100
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Merotocin
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Nolasiban
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Balovaptan
Protein-coding gene in the species Homo sapiens
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin_receptor_1A
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Lipo-oxytocin-1
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
OT-12
Oxytocin receptor antagonist
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Tocinoic_acid
Cleavage product of the arginine vasopressin gene
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Neurophysin_II
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
KNX-101
Vasopressin V1A receptor antagonist
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
RG7713
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Felypressin
G protein-coupled receptor
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin_receptor
Protein-coding gene in the species Homo sapiens
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Vasopressin_receptor_1B
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Relcovaptan
Pharmaceutical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
NMRA-511
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Satavaptan
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
ABT-436
Chemical compound
LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471 V1B Agonists: d[Cha4]AVP DDAVP
Mozavaptan
SRX251
SRX251
SRX251
SRX251
SRX251
SRX251
SRX251
SRX251
SRX251