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PF 184563

  • PF-184563
  • Chemical compound

    PF-184563 is a potent, selective non-peptidic antagonist of the V1a receptor. The compound was discovered by Pfizer in its Sandwich, Kent research center

    PF-184563

    PF-184563

    PF-184563

  • SRX251
  • Pharmaceutical compound

    clinical trials. List of investigational aggression drugs SRX246 Balovaptan PF-184563 Relcovaptan RG7713 "SRX 251". AdisInsight. 3 January 2024. Retrieved 24

    SRX251

    SRX251

    SRX251

  • Tolvaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Tolvaptan

    Tolvaptan

    Tolvaptan

  • Desmopressin
  • Medication

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Desmopressin

    Desmopressin

    Desmopressin

  • Lithium carbonate
  • Chemical compound

    Retrieved 2017-01-02. Yildiz, A; Guleryuz, S; Ankerst, DP; Ongür, D; Renshaw, PF (2008). "Protein kinase C inhibition in the treatment of mania: a double-blind

    Lithium carbonate

    Lithium carbonate

    Lithium_carbonate

  • PF-06655075
  • Pharmaceutical compound

    PF-06655075, also known as PF1 or as ASK1476, is a peripherally selective long-acting peptide oxytocin receptor agonist which is used in scientific research

    PF-06655075

    PF-06655075

  • Vasopressin
  • Mammalian hormone released from the pituitary gland

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin

    Vasopressin

    Vasopressin

  • KNX-100
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    KNX-100

    KNX-100

    KNX-100

  • Cligosiban
  • Pharmaceutical compound

    (INNTooltip International Nonproprietary Name; developmental code names IX-01 and PF-3274167) is an oxytocin receptor antagonist which is or was under development

    Cligosiban

    Cligosiban

    Cligosiban

  • Carbetocin
  • Medication used for preventing postpartum bleeding

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Carbetocin

    Carbetocin

    Carbetocin

  • Vasopressin (medication)
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin (medication)

    Vasopressin (medication)

    Vasopressin_(medication)

  • Oxytocin receptor agonist
  • Chemical compound

    Carbetocin Demoxytocin Lipo-oxytocin-1 (LOT-1) Merotocin (FE-202767) Oxytocin PF-06655075 (PF1; ASK1476) TGOT Vasotocin CA7 – among smallest-known oxytocin

    Oxytocin receptor agonist

    Oxytocin receptor agonist

    Oxytocin_receptor_agonist

  • KNX-101
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    KNX-101

    KNX-101

  • Oxytocin (medication)
  • Medication made from the peptide oxytocin

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Oxytocin (medication)

    Oxytocin (medication)

    Oxytocin_(medication)

  • Oxytocin
  • Peptide hormone and neuropeptide

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Oxytocin

    Oxytocin

    Oxytocin

  • Demeclocycline
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Demeclocycline

    Demeclocycline

    Demeclocycline

  • Barusiban
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Barusiban

    Barusiban

    Barusiban

  • Ornipressin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Ornipressin

    Ornipressin

    Ornipressin

  • Nelivaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Nelivaptan

    Nelivaptan

    Nelivaptan

  • Terlipressin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Terlipressin

    Terlipressin

    Terlipressin

  • LIT-001
  • Small-molecule oxytocin receptor agonist

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    LIT-001

    LIT-001

    LIT-001

  • Vasopressin receptor antagonist
  • Agent that interferes with action at the vasopressin receptors

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin receptor antagonist

    Vasopressin_receptor_antagonist

  • NTX-1472
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    NTX-1472

    NTX-1472

  • SRX246
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    SRX246

    SRX246

    SRX246

  • Atosiban
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Atosiban

    Atosiban

    Atosiban

  • LIT-002
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    LIT-002

    LIT-002

    LIT-002

  • TGOT
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    TGOT

    TGOT

  • Vasotocin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasotocin

    Vasotocin

    Vasotocin

  • Selepressin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Selepressin

    Selepressin

    Selepressin

  • WAY-267464
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    WAY-267464

    WAY-267464

    WAY-267464

  • Uterotonic
  • Medication causing uterine contraction

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Uterotonic

    Uterotonic

  • TC OT 39
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    TC OT 39

    TC OT 39

    TC_OT_39

  • Tocinoic acid
  • Oxytocin receptor antagonist

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Tocinoic acid

    Tocinoic acid

    Tocinoic_acid

  • Retosiban
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Retosiban

    Retosiban

    Retosiban

  • Oxytocin receptor
  • Genes on human chromosome 3

    Carbetocin Demoxytocin Lipo-oxytocin-1 (LOT-1) Merotocin (FE-202767) Oxytocin PF-06655075 (PF1; ASK1476) TGOT Vasotocin CA7 – among smallest-known oxytocin

    Oxytocin receptor

    Oxytocin receptor

    Oxytocin_receptor

  • OT-12
  • Pharmaceutical compound

    literature by Elsa Pflimlin and colleagues by 2020. Oxytocin receptor agonist PF-06655075 (PF1; ASK1476) Pflimlin E, Zhou Z, Amso Z, Fu Q, Lee C, Muppiddi

    OT-12

    OT-12

  • Vasopressin receptor 2
  • Protein-coding gene in the species Homo sapiens

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin receptor 2

    Vasopressin receptor 2

    Vasopressin_receptor_2

  • L-368,899
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    L-368,899

    L-368,899

    L-368,899

  • Demoxytocin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Demoxytocin

    Demoxytocin

    Demoxytocin

  • Brezivaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Brezivaptan

    Brezivaptan

    Brezivaptan

  • Conivaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Conivaptan

    Conivaptan

    Conivaptan

  • Epelsiban
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Epelsiban

    Epelsiban

    Epelsiban

  • Felypressin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Felypressin

    Felypressin

    Felypressin

  • Vasopressin receptor 1B
  • Protein-coding gene in the species Homo sapiens

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin receptor 1B

    Vasopressin receptor 1B

    Vasopressin_receptor_1B

  • WJ0679
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    WJ0679

    WJ0679

    WJ0679

  • Relcovaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Relcovaptan

    Relcovaptan

    Relcovaptan

  • CA7 (drug)
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    CA7 (drug)

    CA7 (drug)

    CA7_(drug)

  • Neurophysin I
  • Cleavage product of the coding protein of OXT gene

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Neurophysin I

    Neurophysin_I

  • NP-1031
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    NP-1031

    NP-1031

  • Vasopressin receptor
  • G protein-coupled receptor

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin receptor

    Vasopressin_receptor

  • Neurophysins
  • Carrier protein for oxytocin and vasopressin

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Neurophysins

    Neurophysins

  • Balovaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Balovaptan

    Balovaptan

    Balovaptan

  • Vasopressin receptor 1A
  • Protein-coding gene in the species Homo sapiens

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Vasopressin receptor 1A

    Vasopressin receptor 1A

    Vasopressin_receptor_1A

  • Nolasiban
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Nolasiban

    Nolasiban

    Nolasiban

  • Lixivaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Lixivaptan

    Lixivaptan

    Lixivaptan

  • RG7713
  • Vasopressin V1A receptor antagonist

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    RG7713

    RG7713

    RG7713

  • Merotocin
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Merotocin

    Merotocin

    Merotocin

  • NMRA-511
  • Pharmaceutical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    NMRA-511

    NMRA-511

  • Neurophysin II
  • Cleavage product of the arginine vasopressin gene

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Neurophysin II

    Neurophysin II

    Neurophysin_II

  • Mozavaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Mozavaptan

    Mozavaptan

    Mozavaptan

  • Satavaptan
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Satavaptan

    Satavaptan

    Satavaptan

  • Lipo-oxytocin-1
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    Lipo-oxytocin-1

    Lipo-oxytocin-1

    Lipo-oxytocin-1

  • L-371,257
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    L-371,257

    L-371,257

    L-371,257

  • ABT-436
  • Chemical compound

    JNJ-17079166 JNJ-17308616 LIT-001 LY-307174 NMRA-511 NTX-1472 (RO-6953958) PF-184563 Relcovaptan RG7713 SRX246 SRX251 TC OT 39 WAY-267464 YM-218 YM-471 YM-35471

    ABT-436

    ABT-436

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