AI & ChatGPT searches , social queries for RO15 4513
Search references for RO15 4513. Phrases containing RO15 4513
See searches and references containing RO15 4513!
Search references for RO15 4513. Phrases containing RO15 4513
See searches and references containing RO15 4513!RO15 4513
Chemical compound
Ro15-4513 is a weak partial inverse agonist of the benzodiazepine class of drugs, developed by Hoffmann–La Roche in the 1980s. It acts as an inverse agonist
Ro15-4513
alpha4beta3delta GABAA receptors are reversed by the behavioral alcohol antagonist Ro15-4513". Proceedings of the National Academy of Sciences of the United States
Short-term effects of alcohol consumption
Short-term_effects_of_alcohol_consumption
Benzodiazepine sedative drug
produced by the α1 subtype of GABAA rather than α5. The inverse agonist Ro15-4513, which blocks the α5 subtype of GABAA, reverses the effects of alcohol
QH-II-66
Agent in biochemistry
effect, whereas inverse agonists have agitation effects (for example, Ro15-4513) or even convulsive and anxiogenic effects (certain beta-carbolines).
Inverse_agonist
Ionotropic receptor and ligand-gated ion channel
lanthanum, riluzole, and menthol. Negative allosteric modulators: flumazenil, Ro15-4513, sarmazenil, pregnenolone sulfate, amentoflavone, and zinc. Inverse allosteric
GABAA_receptor
Pharmacodynamics and pharmacokinetics of ethanol
contribute to ethanol sensitivity. Ro15-4513, a close analogue of the benzodiazepine antagonist flumazenil (Ro15-1788), has been found to bind to the
Pharmacology_of_ethanol
1941 US court case
of the product. No antidote for inebriation was known to science until Ro15-4513 was developed (but not brought to market) in the 1980s. The case name
United_States_v._11_1/4_Dozen_Packages_of_Articles_Labeled_in_Part_Mrs._Moffat's_Shoo-Fly_Powders_for_Drunkenness
6-dihydro-4H-benzo[f]imidazo[1,5-a] [1,4]diazepine-3-carboxylate 3373 78755-81-4 Ro15-4513 ethyl 8-azido-5-methyl-6-oxo-5,6-dihydro-4H-benzo[f]imidazo[1,5-a] [1
List_of_benzodiazepines
Drug class
oenanthotoxin, pentylenetetrazol, phenylsilatrane, picrotoxin, radequinil, Ro15-4513, sarmazenil, suritozole, terbequinil, tetramethylenedisulfotetramine (TETS)
GABAA receptor negative allosteric modulator
GABAA_receptor_negative_allosteric_modulator
Chemical compound
Sarmazenil (Ro15-3505) is a drug from the benzodiazepine family. It acts as a partial inverse agonist of benzodiazepine receptors, meaning that it causes
Sarmazenil
Chemical compound
(GABAA receptors) in the brain. Iomazenil is an analogue of flumazenil (Ro15-1788). 123I-labelled iomazenil can be used to image epileptic seizure foci
Iomazenil
RO15 4513
RO15 4513
RO15 4513
RO15 4513
RO15 4513
RO15 4513
RO15 4513
RO15 4513
RO15 4513