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Chemical compound
Rintodestrant (G1T48) is an orally bioavailable selective estrogen receptor degrader (SERD) discovered in Greg Thatcher's lab at UIC and developed by
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Pharmaceutical company
bladder cancer who are receiving chemotherapy followed by avelumab. Rintodestrant, an oral selective estrogen receptor degrader (SERD), is being developed
G1_Therapeutics
Class of drugs
Sanofi in the lead". Evaluate.com. 2020-02-19. Retrieved 2020-12-28. "Rintodestrant | oral selective estrogen receptor degrader (SERD) | G1 Therapeutics
Selective estrogen receptor degrader
Selective_estrogen_receptor_degrader
estrogen receptor degrader for breast cancer and endometrial cancer Rintodestrant (G1T-48) – selective estrogen receptor modulator and selective estrogen
List of investigational sex-hormonal agents
List_of_investigational_sex-hormonal_agents
Medication for HR+ HER2– breast cancer
ER+/HER2- breast cancer. Studies include palbociclib plus G1 Therapeutic's rintodestrant and Zentalis's Zn-c5. Palbociclib has several direct competitors currently
Palbociclib
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