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CASOPITANT

  • Casopitant
  • Chemical compound

    Casopitant (INNTooltip International Nonproprietary Name), former tentative trade names Rezonic (U.S.) and Zunrisa (Europe), is an NK1 receptor antagonist

    Casopitant

    Casopitant

    Casopitant

  • Aprepitant
  • Chemical compound

    withdrawn. Subsequently, other trials with NK1 receptor antagonists, casopitant and orvepitant, have shown promising results.[needs update] Beyond suggestions

    Aprepitant

    Aprepitant

    Aprepitant

  • NK1 receptor antagonist
  • Chemical compound class

    antiemetic effect in both acute and especially in delayed phases of emesis. Casopitant, netupitant and rolapitant are some newer additions in this group. Rolapitant

    NK1 receptor antagonist

    NK1_receptor_antagonist

  • Antiemetic
  • Drug used to prevent nausea or vomiting

    Aprepitant (Emend) is a commercially available NK1 receptor antagonist Casopitant is an investigational NK1 receptor antagonist Rolapitant (Varubi) another

    Antiemetic

    Antiemetic

  • Tradipitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Tradipitant

    Tradipitant

    Tradipitant

  • Elinzanetant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Elinzanetant

    Elinzanetant

    Elinzanetant

  • Fezolinetant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Fezolinetant

    Fezolinetant

    Fezolinetant

  • Maropitant
  • Veterinary medication

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Maropitant

    Maropitant

    Maropitant

  • Vestipitant
  • Chemical compound

    treatment for tinnitus and insomnia. NK1 receptor antagonist Aprepitant Casopitant Fosaprepitant L-733,060 Maropitant "International Nonproprietary Names

    Vestipitant

    Vestipitant

    Vestipitant

  • Tachykinin receptor 1
  • Protein-coding gene in the species Homo sapiens

    EC50 2nM, 5-amino acid polypeptide chain. CAS# 133156-06-6 Aprepitant Casopitant Elinzanetant Ezlopitant Fosaprepitant Lanepitant Maropitant Rolapitant

    Tachykinin receptor 1

    Tachykinin receptor 1

    Tachykinin_receptor_1

  • Rolapitant
  • Pharmaceutical drug

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Rolapitant

    Rolapitant

    Rolapitant

  • Osanetant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Osanetant

    Osanetant

    Osanetant

  • Substance P
  • Chemical compound (polypeptide neurotransmitter)

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Substance P

    Substance P

    Substance_P

  • Tachykinin peptides
  • Protein family

    veterinary medicine. Examples of tachykinin antagonists include: Aprepitant Casopitant Fosaprepitant Maropitant Nepadutant Osanetant Saredutant Talnetant Tachykinin

    Tachykinin peptides

    Tachykinin peptides

    Tachykinin_peptides

  • List of investigational antidepressants
  • List of pharmaceutical drugs under clinical development for treatment of depression

    (transdermal; BuSpar Patch) – serotonin 5-HT1A receptor partial agonist Casopitant (GW-679769; GW679769) – neurokinin NK1 receptor antagonist Centpropazine

    List of investigational antidepressants

    List_of_investigational_antidepressants

  • Pavinetant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Pavinetant

    Pavinetant

    Pavinetant

  • Netupitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Netupitant

    Netupitant

    Netupitant

  • Burapitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Burapitant

    Burapitant

    Burapitant

  • Lanepitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Lanepitant

    Lanepitant

    Lanepitant

  • ATC code A04
  • Pharmaceutical drug classification

    Metopimazine A04AD10 Dronabinol A04AD11 Nabilone A04AD12 Aprepitant A04AD13 Casopitant A04AD14 Rolapitant A04AD51 Scopolamine, combinations A04AD54 Chlorobutanol

    ATC code A04

    ATC_code_A04

  • List of drugs: C–Ca
  • Casgevy casimersen casirivimab and imdevimab Casodex casokefamide (INN) casopitant (USAN, INN) caspofungin (INN) Casporyn Cassipa Castellani paint Cataflam

    List of drugs: C–Ca

    List_of_drugs:_C–Ca

  • Netupitant/palonosetron
  • Pharmaceutical drug

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Netupitant/palonosetron

    Netupitant/palonosetron

  • Vofopitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Vofopitant

    Vofopitant

    Vofopitant

  • Saredutant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Saredutant

    Saredutant

    Saredutant

  • Talnetant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Talnetant

    Talnetant

    Talnetant

  • Fosaprepitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Fosaprepitant

    Fosaprepitant

    Fosaprepitant

  • Orvepitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Orvepitant

    Orvepitant

    Orvepitant

  • Neurokinin A
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Neurokinin A

    Neurokinin A

    Neurokinin_A

  • Neurokinin B
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Neurokinin B

    Neurokinin B

    Neurokinin_B

  • L-733,060
  • Chemical compound

    in a variety of in vitro models. NK1 receptor antagonists Aprepitant Casopitant Fosaprepitant Maropitant Vestipitant Vofopitant Seabrook GR, Shepheard

    L-733,060

    L-733,060

    L-733,060

  • Tachykinin receptor 3
  • Protein-coding gene in the species Homo sapiens

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Tachykinin receptor 3

    Tachykinin receptor 3

    Tachykinin_receptor_3

  • Ibodutant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Ibodutant

    Ibodutant

    Ibodutant

  • Serlopitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Serlopitant

    Serlopitant

    Serlopitant

  • Nepadutant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Nepadutant

    Nepadutant

    Nepadutant

  • Tachykinin receptor 2
  • Protein-coding gene in the species Homo sapiens

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Tachykinin receptor 2

    Tachykinin receptor 2

    Tachykinin_receptor_2

  • Tachykinin receptor
  • InterPro Family

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Tachykinin receptor

    Tachykinin_receptor

  • Befetupitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Befetupitant

    Befetupitant

    Befetupitant

  • GR-159897
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    GR-159897

    GR-159897

    GR-159897

  • Ezlopitant
  • Chemical compound

    Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant

    Ezlopitant

    Ezlopitant

    Ezlopitant

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