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Chemical compound
Casopitant (INNTooltip International Nonproprietary Name), former tentative trade names Rezonic (U.S.) and Zunrisa (Europe), is an NK1 receptor antagonist
Casopitant
Chemical compound
withdrawn. Subsequently, other trials with NK1 receptor antagonists, casopitant and orvepitant, have shown promising results.[needs update] Beyond suggestions
Aprepitant
Chemical compound class
antiemetic effect in both acute and especially in delayed phases of emesis. Casopitant, netupitant and rolapitant are some newer additions in this group. Rolapitant
NK1_receptor_antagonist
Drug used to prevent nausea or vomiting
Aprepitant (Emend) is a commercially available NK1 receptor antagonist Casopitant is an investigational NK1 receptor antagonist Rolapitant (Varubi) another
Antiemetic
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Tradipitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Elinzanetant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Fezolinetant
Veterinary medication
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Maropitant
Chemical compound
treatment for tinnitus and insomnia. NK1 receptor antagonist Aprepitant Casopitant Fosaprepitant L-733,060 Maropitant "International Nonproprietary Names
Vestipitant
Protein-coding gene in the species Homo sapiens
EC50 2nM, 5-amino acid polypeptide chain. CAS# 133156-06-6 Aprepitant Casopitant Elinzanetant Ezlopitant Fosaprepitant Lanepitant Maropitant Rolapitant
Tachykinin_receptor_1
Pharmaceutical drug
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Rolapitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Osanetant
Chemical compound (polypeptide neurotransmitter)
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Substance_P
Protein family
veterinary medicine. Examples of tachykinin antagonists include: Aprepitant Casopitant Fosaprepitant Maropitant Nepadutant Osanetant Saredutant Talnetant Tachykinin
Tachykinin_peptides
List of pharmaceutical drugs under clinical development for treatment of depression
(transdermal; BuSpar Patch) – serotonin 5-HT1A receptor partial agonist Casopitant (GW-679769; GW679769) – neurokinin NK1 receptor antagonist Centpropazine
List of investigational antidepressants
List_of_investigational_antidepressants
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Pavinetant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Netupitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Burapitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Lanepitant
Pharmaceutical drug classification
Metopimazine A04AD10 Dronabinol A04AD11 Nabilone A04AD12 Aprepitant A04AD13 Casopitant A04AD14 Rolapitant A04AD51 Scopolamine, combinations A04AD54 Chlorobutanol
ATC_code_A04
Casgevy casimersen casirivimab and imdevimab Casodex casokefamide (INN) casopitant (USAN, INN) caspofungin (INN) Casporyn Cassipa Castellani paint Cataflam
List_of_drugs:_C–Ca
Pharmaceutical drug
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Netupitant/palonosetron
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Vofopitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Saredutant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Talnetant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Fosaprepitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Orvepitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Neurokinin_A
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Neurokinin_B
Chemical compound
in a variety of in vitro models. NK1 receptor antagonists Aprepitant Casopitant Fosaprepitant Maropitant Vestipitant Vofopitant Seabrook GR, Shepheard
L-733,060
Protein-coding gene in the species Homo sapiens
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Tachykinin_receptor_3
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Ibodutant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Serlopitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Nepadutant
Protein-coding gene in the species Homo sapiens
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Tachykinin_receptor_2
InterPro Family
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Tachykinin_receptor
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Befetupitant
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
GR-159897
Chemical compound
Agonists: Substance P Antagonists: Aprepitant Befetupitant Burapitant Casopitant CI-1021 CP-96345 CP-99994 CP-122721 Dapitant Elinzanetant Ezlopitant Figopitant
Ezlopitant
CASOPITANT
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CASOPITANT
CASOPITANT
CASOPITANT
CASOPITANT
CASOPITANT
CASOPITANT
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